7-Chloro-2-[3-[[9-(pyridin-4-yl)-3,9-diazaspiro[5.5]undecan-3-yl]carbonyl]phenyl]-2,3-dihydroisoindol-1-one
ELN-441958
CAS: 913064-47-8
Molecular Formula: C29H29ClN4O2
7-Chloro-2-[3-[[9-(pyridin-4-yl)-3,9-diazaspiro[5.5]undecan-3-yl]carbonyl]phenyl]-2,3-dihydroisoindol-1-one - Names and Identifiers
7-Chloro-2-[3-[[9-(pyridin-4-yl)-3,9-diazaspiro[5.5]undecan-3-yl]carbonyl]phenyl]-2,3-dihydroisoindol-1-one - Physico-chemical Properties
| Molecular Formula | C29H29ClN4O2 |
| Molar Mass | 501.02 |
| Solubility | 10 mM in DMSO |
| Storage Condition | 2-8°C |
7-Chloro-2-[3-[[9-(pyridin-4-yl)-3,9-diazaspiro[5.5]undecan-3-yl]carbonyl]phenyl]-2,3-dihydroisoindol-1-one - Preparation solution concentration reference
| 1mg | 5mg | 10mg | |
|---|---|---|---|
| 1 mM | 1.996 ml | 9.98 ml | 19.959 ml |
| 5 mM | 0.399 ml | 1.996 ml | 3.992 ml |
| 10 mM | 0.2 ml | 0.998 ml | 1.996 ml |
| 5 mM | 0.04 ml | 0.2 ml | 0.399 ml |
Last Update：2024-01-02 23:10:35
7-Chloro-2-[3-[[9-(pyridin-4-yl)-3,9-diazaspiro[5.5]undecan-3-yl]carbonyl]phenyl]-2,3-dihydroisoindol-1-one - Reference Information
| biological activity | ELN-441958 is a potent B1 receptor antagonist, inhibition of the B1 agonist ligand [3H] DAKD binds to IMR-90 cells with a Ki of 0.26 nM. Inhibition of the B1 receptor in ELN-441958 is more selective than inhibition of the B2 receptor, the selectivity was more than 500 and 2000 fold higher than inhibition of μ/δ opioid receptors, respectively. |
Last Update：2024-04-09 21:21:28
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Product Name: ELN-441958 Visit Supplier Webpage Request for quotation
CAS: 913064-47-8
Tel: 18301782025
Email: 3008007409@qq.com
Mobile: 18021002903
QQ: 3008007409
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CAS: 913064-47-8
Tel: 18301782025
Email: 3008007409@qq.com
Mobile: 18021002903
QQ: 3008007409
Wechat: 18301782025
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